H-151 is a potent, irreversible, and selective small-molecule inhibitor of STING [1], a key sensor of cytosolic nucleic acids. STING is a transmembrane ...
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Xếp hạng 5,0 (10) H-151 is a potent, selective and covalent antagonist of STING that has noteworthy inhibitory activity both in cells and in vivo. H-151 reduces TBK1 ...
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Xếp hạng 5,0 (9) H-151 is a highly potent and covalent antagonist of STING that has noteworthy inhibitory activity both in human cells and in vivo. Targets. STING. In vivo.
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H-151 displayed anti-inflammatory activity in both keratinocytes and immune cells, and decreased the severity of psoriatic response in vivo.
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H 151 is a STING antagonist. Covalently binds STING at Cys91, blocking palmitoylation and preventing assembly of STING clusters. Decreases inflammatory cytokine ...
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H-151 is an inhibitor of stimulator of interferon genes (STING). ... It forms an adduct with mouse STING in serum and acts in an irreversible manner. It inhibits ...
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25,00 SGD Còn hàng Shop H151 Headset. Features in-line controls for volume and to mute calls, rotating noise cancelling microphone, adjustable headband, and 3.5mm audio jack.
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Comment: H-151 is a small molecule covalent STING antagonist [2]. Mechanistically it binds to Cys91 of the protein and prevents its palmitoylation.
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H 151 is a STING antagonist. Covalently binds STING at Cys91, blocking palmitoylation and preventing assembly of STING clusters.
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8 thg 4, 2021 · H151 is a covalent small molecule inhibiting STING palmitoylation and thus blocking STING-mediated signaling pathways. H151 was identified as a ...
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7 thg 6, 2021 · The most promising reported STING antagonist, H-151, is a covalent inhibitor that binds to a reactive Cys91 in the transmembrane domain of STING ...
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View and buy high purity H 151 from Tocris Bioscience, a Bio-Techne brand. STING antagonist.
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Xếp hạng 5,0 (1) H-151 ≥98% (HPLC); CAS Number: 941987-60-6; Synonyms: 1-(4-Ethylphenyl)-3-(1H-indol-3-yl) urea; find Sigma-Aldrich-SML2437 MSDS, related peer-reviewed ...
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H-151 is a potent and irreversible inhibitor of stimulator of interferon genes (STING). It covalently modifies cysteine 91 of STING, which blocks STING ...
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